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受託サービス

バインディングアッセイサービス

概要

RIを用いるバンディングアッセイはレセプターの結合アッセイなど、歴史も長く、化合物の薬理活性を確実に評価する方法として確立しています。レセプターとしてラット由来のもの、あるいはヒト型レセプターなどがあり、目的に合わせて使い分けることができます。弊社ではキャリパーライフサイエンス社のラボラトリーオートメーション技術をフルに活用した、安心、確実なデータをご提供するアッセイシステムを構築し、活用しています。

 

得られたデータは社内のQA基準に従って評価をし、お客様には信頼性の高いデータをご提供します。

 

また、弊社ではSOPの整備をはじめ、アッセイを管理する様々な仕組みが整っています。お客様のサンプルのアッセイをGLPに準拠したやり方で進めることも可能となっていますので、お客様の様々な御要望に応じることが可能です。詳しくはお問合せください。

 

下表は、バインディングアッセイの2010年6月現在の表です。最新版の価格は米国のWEBサイトを参照してください。

Cat# Assay Type Assay Class Assay Name
100-0001 Binding Adenosine Transporter AOT (h)
100-0003 Binding Adenosine A2A (h)
100-0004 Binding Adenosine A3
100-0005 Binding Adrenergic Alpha 1A
100-0006 Binding Adrenergic Alpha 1B
100-0007 Binding Adrenergic Alpha 2A (h)
100-0008 Binding Adrenergic Alpha 2B
100-0009 Binding Adrenergic Alpha 2C (h)
100-0010 Binding Adrenergic Beta 1 (h)
100-0011 Binding Adrenergic Beta 2 (h)
100-0012 Binding Bradykinin B2
100-0013 Binding Calcium Type L (Dihydropyridine Site)
100-0014 Binding Calcium Type N
100-0015 Binding Dopamine Transporter, DAT
100-0016 Binding Dopamine D1 (h)
100-0018 Binding Dopamine D3
100-0019 Binding Dopamine D4.4 (h)
100-0021 Binding GABA GABA-A Agonist Site
100-0022 Binding GABA GABA-A BDZ Alpha-1 Site
100-0023 Binding GABA Chloride TBOB Site
100-0024 Binding GABA-B GABA-B
100-0026 Binding Glutamate AMPA Site
100-0027 Binding Glutamate Kainate Site
100-0028 Binding Glutamate NMDA MK801 Site
100-0029 Binding Glutamate NMDA Agonist Site
100-0030 Binding Adenosine AD Non selective
100-0031 Binding Glutamate NMDA PCP Site
100-0032 Binding Glutamate NMDA Glycine Strychnine-insensitive
100-0033 Binding Glycine Glycine Strychnine-sensitive Site
100-0034 Binding Histamine H1
100-0035 Binding Histamine H3
100-0036 Binding Leukotriene LTB4 (BLT)
100-0037 Binding Leukotriene LTD4 (CysLT1)
100-0038 Binding Muscarinic M1 (h)
100-0039 Binding Muscarinic M2 (h)
100-0040 Binding Muscarinic M3 (h)
100-0041 Binding Muscarinic M4 (h)
100-0042 Binding Muscarinic M5 (h)
100-0043 Binding Adenosine A2
100-0044 Binding Neurokinin NK1
100-0045 Binding Neuropeptide Y NPY2 (h)
100-0046 Binding Nicotinic a-BnTx Insensitive Neuronal
100-0047 Binding Adenosine Transporter AOT
100-0048 Binding Norepinephrine Transporter NET
100-0049 Binding Opioid Delta-2 (h)
100-0051 Binding Opioid Mu (h)
100-0052 Binding Potassium ATP Sensitive (KATP)
100-0054 Binding Potassium Ca2+ Activated (VI)
100-0055 Binding Purinergic P2Y (h)
100-0056 Binding Serotonin Transporter SERT
100-0057 Binding Serotonin 5HT1A (h)
100-0058 Binding Serotonin 5HT1D
100-0059 Binding Serotonin 5HT2A
100-0060 Binding Serotonin 5HT2C
100-0061 Binding Serotonin 5HT3
100-0062 Binding Serotonin 5HT4
100-0063 Binding Serotonin 5HT5A (h)
100-0064 Binding Serotonin 5HT6 (h)
100-0065 Binding Serotonin 5HT7 (h)
100-0066 Binding Sigma S1
100-0067 Binding Sigma S2
100-0069 Binding Sodium Site 2
100-0070 Binding Thromboxane TXA2 (h)
100-0072 Binding Opioid Nociceptin, ORL1 (h)
100-0073 Binding Cannabinoid CB1 (h)
100-0074 Binding Cannabinoid CB2 (h)
100-0075 Binding Imidazoline I2 central
100-0084 Binding Angiotensin II AT1 (h)
100-0085 Binding Endothelin ETA (h)
100-0086 Binding Histamine H2
100-0089 Binding Nitric Oxide NOS (neuronal-binding)
100-0099 Binding Serotonin Transporter SERT (h)
100-0100 Binding Adrenergic Alpha 1 Non selective
100-0101 Binding Adrenergic Alpha 2 Non selective
100-0102 Binding Adrenergic Alpha 2C
100-0103 Binding Adrenergic Beta Non selective
100-0104 Binding Adrenergic Beta 1
100-0105 Binding Adrenergic Beta 2
100-0106  Binding  Adenylate Cyclase  Forskolin 
100-0107 Binding Angiotensin II AT1 Peripheral
100-0108 Binding Angiotensin II AT2 Central
100-0109 Binding Atrial Naturietic Factor ANP-A
100-0110 Binding Benzodiazepine (peripheral) Mitochondrial Translocator Protein (TSPO)
100-0111 Binding Benzodiazepine (peripheral) Mitochondrial Translocator Protein (TSPO) (h)
100-0113 Binding Calcium Type L (Benzothiazepine Site)
100-0114 Binding Cholecystokinin CCKA
100-0115 Binding Cholecystokinin CCKB
100-0116 Binding Dopamine DA Non-Selective (Clozapine)
100-0117 Binding Complement Anaphylatoxin C5aR (h)
100-0118 Binding Corticotropin Releasing Factor CRF Non selective
100-0120 Binding Dopamine D1
100-0121 Binding Dopamine D2
100-0123 Binding Dopamine Transporter, DAT (h)
100-0124 Binding Endothelin ETB (h)
100-0125 Binding Epidermal Growth Factor EGF
100-0129 Binding GABA GABA-A BDZ Alpha-6 Site
100-0130 Binding Galanin Galanin Non selective
100-0131 Binding Glutamate Chloride Dependent Site
100-0132 Binding Imidazoline I1 peripheral
100-0133 Binding Inositol Triphosphate IP3
100-0134 Binding Melatonin Melatonin Non selective
100-0135 Binding Muscarinic M Non selective Central
100-0136 Binding Muscarinic M Non selective Peripheral
100-0137 Binding Muscarinic M1
100-0138 Binding Muscarinic M2
100-0139 Binding Muscarinic M3
100-0140 Binding Neurokinin NK2 (NKA) (h)
100-0141 Binding Neurokinin NK3 (NKB)
100-0142 Binding Neuropeptide Y NPY Non selective
100-0143 Binding Neuropeptide Y NPY1 (h)
100-0144 Binding Neurotensin NT
100-0145 Binding Neurotensin NT (h)
100-0146 Binding Norepinephrine Transporter NET (h)
100-0147 Binding Opioid OP Non-selective
100-0148 Binding Opioid OP Non-selective (+Na+)
100-0149 Binding Opioid Delta
100-0150 Binding Opioid Kappa 1
100-0151 Binding Opioid Mu
100-0152 Binding Oxytocin Oxytocin
100-0153 Binding Platelet Activating Factor PAF
100-0154 Binding Progesterone Progesterone (bov)
100-0155 Binding Progesterone Progesterone (h)
100-0156 Binding Protein Kinase C PDBu
100-0157 Binding Purinergic P2Y
100-0158 Binding Serotonin 5HT Non selective
100-0159 Binding Serotonin 5HT1 Non selective
100-0160 Binding Serotonin 5HT1A
100-0161 Binding Serotonin 5HT1B
100-0162 Binding Serotonin 5HT1D (h)
100-0163 Binding Serotonin 5HT2A (h)
100-0164 Binding Sigma S Non selective
100-0165 Binding Somatostatin SOM Non selective
100-0166 Binding Testosterone (Androgen) Testosterone Cytosolic (rat)
100-0167 Binding Testosterone (Androgen) Testosterone Cytosolic (h)
100-0168 Binding Testosterone (Androgen) Testosterone Nuclear
100-0169 Binding Thyrotropin Releasing Hormone TRH
100-0170 Binding Vasoactive Intestinal Peptide VIP Non selective
100-0171 Binding Vasopressin V1
100-0172 Binding Vasopressin V1A (h)
100-0325 Binding Adrenergic Beta 3 (h)
100-0328  Binding  Adenosine  A1 (h) 
100-0329 Binding GABA GABA Non selective
100-0330 Binding Potassium hERG (I[Kr]) (h)
100-0333  Binding  Calcium  Type L (a2d Subunit) 
100-0359 Binding Nicotinic a-BnTx Insensitive Neuronal (h)
100-0403 Binding Nicotinic a-BnTx Sensitive Muscle-Type (h)
100-0405 Binding Glutamate (metabotropic) mGluR5
100-0406 Binding Serotonin 5HT3 (h)
100-0408 Binding Tumor Necrosis Factor TNFa (h)
100-0448 Binding Glucocorticoid Glucocorticoid (h)
100-0456 Binding Histamine H1 (h)
100-0481 Binding Leukotriene LTB4 (BLT1) (h)
100-0482 Binding Leukotriene LTB4 (BLT2) (h)
100-0751 Binding Vesicular Monoamine Transporter VMAT2
100-0756 Binding Glutamate (metabotropic) mGluR1
100-0786 Binding GammaHydroxyButyrate GHB
100-0806 Binding P-Glyocoprotein (PGP) Transporter P-Glycoprotein (PGP) (h)
100-0848 Binding Serotonin 5HT2B (h)
100-0872 Binding Retinoic Acid Retinoic Acid Receptor, RARa (h) Agonist Binding
100-0877 Binding Retinoic Acid Retinoic Acid Receptor (h) Antagonist Binding
100-0887 Binding Opioid Nociceptin, ORL1 brain (rat)
100-0888 Binding Opioid Nociceptin, ORL1 brain (h)
100-0889 Binding Opioid Nociceptin, ORL1 brain (macaque)
100-0893 Binding Mineralocorticoid Mineralocorticoid (rat)
100-0911 Binding Farnesoid Farnesoid X Receptor (h), Antagonist
100-0912  Binding  Farnesoid  Farnesoid X Receptor (h), Agonist 
100-0913 Binding Retinoic Acid Retinoic Acid Receptor (rat)
100-0971 Binding Nicotinic α-Bungarotoxin Sensitive, Neuronal (α7)
100-0990 Binding Adrenergic Alpha2b (h)
100-1005 Binding Dopamine D4.2 (h)
100-1006 Binding Dopamine D2s (h)
100-1024 Binding Opioid Nociceptin, ORL1 brain (Rabbit)